Slow, tight-binding inhibition of PDF by actinonin induces
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Peptide Deformylase as an Antibacterial Drug Target: Target Validation and Resistance Development
Frédéric Dardel's research works Paris Descartes University, Paris and other places
Aminopeptidase inhibitors bestatin and actinonin inhibit cell proliferation of myeloma cells predominantly by intracellular interactions - ScienceDirect
Trapping Conformational States Along Ligand-Binding Dynamics of Peptide Deformylase: The Impact of Induced Fit on Enzyme Catalysis
JCM, Free Full-Text
3D comparison of the binding between various PDFIs and actinonin.: (a)
/articles/PMC6759494/bin/nihms-104982
Carmela GIGLIONE, Laboratory Head, PhD, Université Paris-Saclay, Paris
6: Slow Binding Inhibitors
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